Molecule Details
InChIKeyCYBHYVCTXZJLET-UHFFFAOYSA-N
Compound Name17-Oxo-2-oxa-9,11,15,18-tetrazapentacyclo[17.6.2.13,7.09,13.023,27]octacosa-1(26),3,5,7(28),10,12,19,21,23(27),24-decaene-4-carbonitrile
Canonical SMILESN#Cc1ccc2cc1Oc1ccc3cccc(c3c1)NC(=O)CNCc1cncn1C2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.64
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.4 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.4 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 6.2 IC50 ChEMBL