Molecule Details
InChIKeyCXNXFUAHKZOVID-UHFFFAOYSA-N
Compound Namen-[5-(1,1-Dioxo-1lambda6-isothiazolidin-2-yl)-1h-indazol-3-yl]-2-[4-(methylsulfonyl)phenyl]acetamide
Canonical SMILESCS(=O)(=O)c1ccc(CC(=O)Nc2n[nH]c3ccc(N4CCCS4(=O)=O)cc23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 7.7 pIC50 TTD_MultiTarget
P06493 CDK1 Homo sapiens Human PF00069 7.2 pIC50 TTD_MultiTarget
P11802 CDK4 Homo sapiens Human PF00069 7.2 pIC50 TTD_MultiTarget