Molecule Details
InChIKeyCXIDTYUJLXWEAY-UHFFFAOYSA-N
Compound Name5-[3-[4-(2,5-Dimethylphenyl)piperazin-1-yl]-3-oxopropyl]-5-pyridin-2-ylimidazolidine-2,4-dione
Canonical SMILESCc1ccc(C)c(N2CCN(C(=O)CCC3(c4ccccn4)NC(=O)NC3=O)CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P78536 ADAM17 Homo sapiens Human PF16698 PF00200 PF13574 6.9 IC50 ChEMBL;BindingDB
Q9UNA0 ADAMTS5 Homo sapiens Human PF17771 PF19236 PF05986 PF01421 PF19030 PF00090 6.9 IC50 ChEMBL;BindingDB