Molecule Details
InChIKeyCXCXNZWXDOVZBA-UHFFFAOYSA-N
Compound Name7-Cyclopentyl-2-({1-Methyl-5-[(4-Methylpiperazin-1-Yl)carbonyl]-1h-Pyrrol-3-Yl}amino)-7h-Pyrrolo[2,3-D]pyrimidine-6-Carboxamide
Canonical SMILESCN1CCN(C(=O)c2cc(Nc3ncc4cc(C(N)=O)n(C5CCCC5)c4n3)cn2C)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P06493 CDK1 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB