Molecule Details
InChIKeyCWYCYSJSUHLIBI-LJAQVGFWSA-N
Compound Name5-[4-(2-phenylphenyl)piperazin-1-yl]-1-[(2S)-2-(piperidine-1-carbonyl)pyrrolidin-1-yl]pentan-1-one
Canonical SMILESO=C([C@@H]1CCCN1C(=O)CCCCN1CCN(c2ccccc2-c2ccccc2)CC1)N1CCCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P34969 HTR7 Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB
P50406 HTR6 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB