Molecule Details
InChIKeyCVNQRFZZFGTWIK-UHFFFAOYSA-N
Compound Name1-[2-[[5-fluoro-4-[7-fluoro-2-methyl-3-(4-methylcyclohexyl)benzimidazol-5-yl]pyrimidin-2-yl]amino]-7,8-dihydro-5H-1,6-naphthyridin-6-yl]-2-(methylamino)ethanone
Canonical SMILESCNCC(=O)N1CCc2nc(Nc3ncc(F)c(-c4cc(F)c5nc(C)n(C6CCC(C)CC6)c5c4)n3)ccc2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 8.6 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB