Molecule Details
InChIKeyCVKTUICDKSUYDI-UHFFFAOYSA-N
Compound NameN6-[(2,5-dimethoxyphenyl)methyl]pyrido[2,3-d]pyrimidine-2,4,6-triamine
Canonical SMILESCOc1ccc(OC)c(CNc2cnc3nc(N)nc(N)c3c2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.07
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00381 folA Lacticaseibacillus casei Pathogen PF00186 7.8 IC50 ChEMBL;BindingDB
B0BL08 dfrA17 Escherichia coli Pathogen PF00186 6.9 IC50 BindingDB
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 6.5 IC50 ChEMBL;BindingDB