Molecule Details
InChIKeyCVCDJFWPDDHHOS-IURJAOHMSA-N
Canonical SMILESCCCC[C@H](NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CNC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccc(S(=O)(=O)O)cc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)OCCc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P04746 AMY2A Homo sapiens Human PF00128 PF02806 9.5 IC50 ChEMBL;BindingDB
P32239 CCKBR Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB