Molecule Details
InChIKeyCUSUZSREAOLZQQ-ZZXKWVIFSA-N
Compound Name(E)-N-[4-(morpholin-4-ylmethyl)phenyl]-3-[4-(1H-pyrazol-4-yl)-3-pyridinyl]prop-2-enamide
Canonical SMILESO=C(/C=C/c1cnccc1-c1cn[nH]c1)Nc1ccc(CN2CCOCC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 9.3 IC50 ChEMBL;BindingDB
P49336 CDK8 Homo sapiens Human PF00069 9.3 IC50 ChEMBL
Q9BWU1 CDK19 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB