Molecule Details
InChIKeyCUMVKGYWZJOYNO-UHFFFAOYSA-N
Compound Name8-(2,6-Dimethylpyridin-4-yl)-7-(4-fluoropheny1)-2-[(3-fluoropyridin-2-yl)methyl]-[l,2,4]triazolo [1,5-c]pyrimidin-5-amine
Canonical SMILESCn1cc(-c2c(-c3ccc(F)cc3)nc(N)n3nc(Cc4ncccc4F)nc23)ccc1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB