Molecule Details
InChIKeyCTXDQIFHYWGFBV-CONSDPRKSA-N
Canonical SMILESCOc1cccc(CCNC(=O)C[C@H](O)[C@H](COCc2ccc(-c3ccccc3)cc2)NC(=O)c2c(F)cc(F)cc2F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P39898 PMI Plasmodium falciparum (isolate HB3) Pathogen PF00026 6.9 Ki ChEMBL;BindingDB
P46925 PMII Plasmodium falciparum (isolate HB3) Pathogen PF00026 6.5 Ki ChEMBL;BindingDB