Molecule Details
InChIKeyCTVCNKIVQXSUSH-UHFFFAOYSA-N
Canonical SMILESCc1ccc(N2Cc3c(nc(C)c(CN)c3-c3ccc(Cl)cc3Cl)C2=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P27487 DPP4 Homo sapiens Human PF00930 PF00326 7.9 Ki ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.6 IC50 ChEMBL;BindingDB