Molecule Details
InChIKeyCTSPAMFJBXKSOY-UHFFFAOYSA-N
Canonical SMILESCc1c2ccncc2c(C)c2c1[nH]c1ccccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB17026
Drug NameEllipticine
CAS Number519-23-3
Groups experimental
ATC Codes nan
DescriptionEllipticine is a potent antineoplastic agent.[A252992]

Categories: Alkaloids Antineoplastic Agents Carbazoles Enzyme Inhibitors Heterocyclic Compounds, Fused-Ring Indole Alkaloids Indoles Indolizidines Indolizines Secologanin Tryptamine Alkaloids Uncoupling Agents
Cross-references: BindingDB: 50004233 ChEBI: 4776 CHEMBL123 ChemSpider: 3100 C09154 Wikipedia: Ellipticine ZINC: ZINC000001846592
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P04798 CYP1A1 Homo sapiens Human PF00067 7.7 IC50 ChEMBL;BindingDB
P10721 KIT Homo sapiens Human PF00047 PF07714 6.7 IC50 ChEMBL
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P11388 TOP2A DNA topoisomerase 2-alpha inhibitor targets
Q02880 TOP2B DNA topoisomerase 2-beta inhibitor targets