Molecule Details
InChIKeyCTDCQQXDSZWWIE-HRAATJIYSA-N
Compound NameN-[4-[(2S,5S)-2-(6-amino-3-pyridinyl)-5-methylmorpholin-4-yl]butyl]-1H-indole-2-carboxamide
Canonical SMILESC[C@H]1CO[C@@H](c2ccc(N)nc2)CN1CCCCNC(=O)c1cc2ccccc2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB