Molecule Details
InChIKeyCSTRIVMEIYPLGJ-ASUDMDKOSA-N
Canonical SMILESCc1cc(-c2nc(NC[C@H]3CCC[C@@H](c4ccc(C(F)(F)F)cc4)O3)c(C)c(C(=O)N3CCC(N[C@@H]4CCOC[C@@H]4F)CC3)n2)no1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41597 CCR2 Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P51681 CCR5 Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB