Molecule Details
InChIKeyCSSQSFDPFAFVFE-UHFFFAOYSA-N
Compound Name4$#8243;-methyl-5''-sulfamoyl-4''-(2H-tetrazol-5-yl)-[1,1'':3'',1$#8243;-terphenyl]-4-carboxamide
Canonical SMILESCc1ccc(-c2cc(-c3ccc(C(N)=O)cc3)cc(S(N)(=O)=O)c2-c2nn[nH]n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.79
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.2 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 7.3 IC50 BindingDB
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 6.9 IC50 BindingDB