Molecule Details
InChIKeyCSNKQXLBFBGYCU-HNNXBMFYSA-N
Compound Name(3S)-1-[6-[1-methyl-5-(1-methylpyrazol-4-yl)pyrazolo[3,4-c]pyridin-3-yl]-2-pyridinyl]piperidin-3-amine
Canonical SMILESCn1cc(-c2cc3c(-c4cccc(N5CCC[C@H](N)C5)n4)nn(C)c3cn2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.6 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.4 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.8 Ki ChEMBL;BindingDB