Molecule Details
InChIKeyCSIWGLJKPPOVQR-UHFFFAOYSA-N
Compound NamePyrazoloquinazoline deriv., 17
Canonical SMILESCOc1cc2c(Nc3cc(CC(=O)Nc4cccc(C(F)(F)F)c4)[nH]n3)ncnc2cc1OCCCN1CCC(CO)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.36
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75716 STK16 Homo sapiens Human PF00069 7.9 pIC50 TTD_MultiTarget
O14965 AURKA Homo sapiens Human PF00069 7.1 Ki ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 7.1 Ki ChEMBL;BindingDB