Molecule Details
InChIKeyCSFNNUIZTRGKSQ-UHFFFAOYSA-N
Compound NameN-(3-{4-[1-Ethyl-3-(4-{[(phenylamino)carbonyl]amino}phenyl)-1H-pyrazol-4-yl]-1H-pyrrolo[2,3-b]pyridin-2-yl}phenyl)acetamide
Canonical SMILESCCn1cc(-c2ccnc3[nH]c(-c4cccc(NC(C)=O)c4)cc23)c(-c2ccc(NC(=O)Nc3ccccc3)cc2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.05
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.9 pIC50 TTD_MultiTarget