Molecule Details
InChIKeyCSBKUBOVPUXFLO-MAVVKCOWSA-N
Canonical SMILESCO[C@H]1CC[C@H](CNc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CC(C)(C)CC5)CC4)cc3Oc3cnc4[nH]ccc4c3)cc2[N+](=O)[O-])CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P10415 BCL2 Homo sapiens Human PF00452 PF02180 11.0 Ki ChEMBL;BindingDB
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 7.8 Ki ChEMBL;BindingDB
Q92843 BCL2L2 Homo sapiens Human PF00452 PF02180 6.1 Ki ChEMBL