Molecule Details
InChIKeyCRWXJGJNJZPMRW-UHFFFAOYSA-N
Compound Namen-(4-Bromo-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(2-oxo-6-(trifluoromethyl)quinolin-1(2h)-yl)acetamide
Canonical SMILESO=C(Cn1c(=O)ccc2cc(C(F)(F)F)ccc21)Nc1scc(Br)c1-c1ncn[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.35
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB