Molecule Details
InChIKeyCRVXXEZDJABOJD-UHFFFAOYSA-N
Compound Name7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]-1H-quinolin-2-one
Canonical SMILESCOc1ccccc1N1CCN(CCCCOc2ccc3ccc(=O)[nH]c3c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 9.8 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB