Molecule Details
InChIKeyCRHLQSKLPOQEER-UHFFFAOYSA-N
Compound Name7-(4-(4-o-tolylpiperazin-1-yl)butoxy)-3,4-dihydro-1,8-naphthyridin-2(1H)-one
Canonical SMILESCc1ccccc1N1CCN(CCCCOc2ccc3c(n2)NC(=O)CC3)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.0
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB