Molecule Details
InChIKeyCQRFXINTEFATOH-OAHLLOKOSA-N
Compound Name(3R)-1-[2-amino-6-(3-amino-1H-indazol-6-yl)pyrimidin-4-yl]-N-phenylpiperidine-3-carboxamide
Canonical SMILESNc1nc(-c2ccc3c(N)n[nH]c3c2)cc(N2CCC[C@@H](C(=O)Nc3ccccc3)C2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.9
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O15530 PDPK1 Homo sapiens Human PF14593 PF00069 6.9 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 Clinical TTD_MultiTarget TTD_MultiTarget