Molecule Details
InChIKeyCQOOBCLBMYGVDE-UHFFFAOYSA-N
Compound Name2-cyclopentyl-N-(3-(4-((1-methylpiperidin-4-yl)oxy)phenyl)-1H-indazol-5-yl)-2-(pyridin-2-yl)acetamide
Canonical SMILESCN1CCC(Oc2ccc(-c3n[nH]c4ccc(NC(=O)C(c5ccccn5)C5CCCC5)cc34)cc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33981 TTK Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 7.2 IC50 ChEMBL
Q9NQS7 INCENP Homo sapiens Human PF03941 PF12178 7.2 IC50 ChEMBL