Molecule Details
InChIKeyCQHOSPMLVTXHPG-UHFFFAOYSA-N
Compound Name4-{2-methylimidazo[1,2-a]pyridin-3-yl}-N-phenylpyrimidin-2-amine
Canonical SMILESCc1nc2ccccn2c1-c1ccnc(Nc2ccccc2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.44
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.4 pIC50 TTD_MultiTarget
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 7.4 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.4 pIC50 TTD_MultiTarget