Molecule Details
InChIKeyCPKUIKQUAANRIQ-UHFFFAOYSA-N
Compound Name1-benzyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
Canonical SMILESO=S(=O)(c1cccc2ccccc12)c1nn(Cc2ccccc2)c2ccc(N3CCNCC3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.06
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P50406 HTR6 Homo sapiens Human PF00001 8.1 IC50 ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB