Molecule Details
InChIKeyCOYPPYFVEXHGJK-UHFFFAOYSA-N
Compound Name5-Chloro-2-[1-(4-chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-1H-benzoimidazole
Canonical SMILESClc1ccc(CN2CC=C(c3nc4cc(Cl)ccc4[nH]3)CC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB