Molecule Details
InChIKeyCOTQDURISRILOR-CQSZACIVSA-L
Compound Name2-[5-[2-(ethylcarbamoylamino)-6-fluoro-7-[(2R)-oxolan-2-yl]-3H-benzimidazol-5-yl]pyrimidin-2-yl]propan-2-yl phosphate
Canonical SMILESCCNC(=O)Nc1nc2cc(-c3cnc(C(C)(C)OP(=O)([O-])[O-])nc3)c(F)c([C@H]3CCCO3)c2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P0A0K8 gyrB Staphylococcus aureus Pathogen PF00204 PF00986 PF02518 PF01751 7.3 IC50 ChEMBL;BindingDB
P0C1S7 parE Staphylococcus aureus Pathogen PF00204 PF00986 PF02518 PF01751 7.2 IC50 ChEMBL