Molecule Details
InChIKeyCOBLQYUYOHSZOW-UHFFFAOYSA-N
Compound NameN-[3-[(4-Fluoro-1-piperidinyl)methyl]-5-isothiazolyl]-6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-amine Hydrochloride
Canonical SMILESCc1cn2c(-c3cn[nH]c3)cnc2c(Nc2cc(CN3CCC(F)CC3)ns2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.74
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O75716 STK16 Homo sapiens Human PF00069 8.4 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB