Molecule Details
InChIKeyCOANUJWURZDRKT-UHFFFAOYSA-N
Compound Name4-[[3-(Dimethylamino)-1-[5-[(2-fluorobenzoyl)amino]cyclohexa-1,5-dien-1-yl]propyl]amino]quinazoline-8-carboxamide
Canonical SMILESCN(C)CCC(Nc1ncnc2c(C(N)=O)cccc12)C1=CCCC(NC(=O)c2ccccc2F)=C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 7.7 IC50 ChEMBL;BindingDB