Molecule Details
InChIKeyCNWXJSZWVGJITL-HECCNADXSA-N
Compound Namedeamino-Tyr(SO3H)-Nle-Gly-Trp-N(Me)Leu-Asp-Phe-NH2
Canonical SMILESCCCC[C@H](NC(=O)CCc1ccc(OS(=O)(=O)O)cc1)C(=O)NCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N(C)[C@@H](CC(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.62
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 9.6 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 9.6 IC50 ChEMBL;BindingDB