Molecule Details
InChIKeyCNWAVQYSQHXMCH-UHFFFAOYSA-N
Compound Name4-(4-amino-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2,6-difluorobenzaldehyde
Canonical SMILESCC(C)n1nc(-c2cc(F)c(C=O)c(F)c2)c2c(N)ncnc21
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.18
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08631 HCK Homo sapiens Human PF07714 PF00017 PF00018 6.3 IC50 ChEMBL
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 6.1 IC50 ChEMBL
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.1 pIC50 TTD_MultiTarget