Molecule Details
InChIKeyCNVDRXITZNMNTP-APPZFPTMSA-N
Compound Name8-bromo-2-[(2S,4R)-4-hydroxypyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3H)-one
Canonical SMILESO=c1[nH]c([C@@H]2C[C@@H](O)CN2)nc2c1oc1ccc(Br)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL6.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
O00311 CDC7 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P67870 CSNK2B Homo sapiens Human PF01214 6.4 IC50 ChEMBL
P68400 CSNK2A1 Homo sapiens Human PF00069 6.4 IC50 ChEMBL