Molecule Details
InChIKeyCMMQUPMVPKKYRI-UHFFFAOYSA-N
Compound Name6-(2-aminoethylsulfonyl)-3-(2-methyl-1H-benzimidazol-4-yl)-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESCc1nc2c(-c3ccc(S(=O)(=O)CCN)c(S(N)(=O)=O)c3-c3nn[nH]n3)cccc2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.68
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.8 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.7 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.5 IC50 BindingDB