Molecule Details
InChIKeyCMGCUKSVHPVYFF-UHFFFAOYSA-N
Compound Name1-[3-[[1-[2-(2-Methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]phenyl]pyrrolidin-2-one
Canonical SMILESCc1ccc2c(OCCN3CCC(Cc4cccc(N5CCCC5=O)c4)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.2
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB