Molecule Details
InChIKeyCLZRGXQPCQFFTL-NHPFZIKMSA-N
Compound Name(2S)-N-[(2S)-3-(cyclopenten-1-yl)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]-3-(4-methoxyphenyl)-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide
Canonical SMILESCOc1ccc(C[C@H](NC(=O)[C@H](C)NC(=O)CN2CCOCC2)C(=O)N[C@@H](CC2=CCCC2)C(=O)[C@@]2(C)CO2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28062 PSMB8 Homo sapiens Human PF00227 7.1 IC50 ChEMBL;BindingDB
P28065 PSMB9 Homo sapiens Human PF00227 6.7 IC50 ChEMBL;BindingDB
P28074 PSMB5 Homo sapiens Human PF00227 6.0 IC50 ChEMBL;BindingDB