Molecule Details
InChIKeyCLHZIKCWBUWLQU-UHFFFAOYSA-N
Compound Name2-benzylsulfonyl-N-[2-(cyclopropylamino)-2-oxoethyl]-2-[6-(6-fluoro-3-pyridinyl)-1,3-benzothiazol-2-yl]acetamide
Canonical SMILESO=C(CNC(=O)C(c1nc2ccc(-c3ccc(F)nc3)cc2s1)S(=O)(=O)Cc1ccccc1)NC1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11150 LIPC Homo sapiens Human PF00151 PF01477 8.2 IC50 ChEMBL;BindingDB
Q9Y5X9 LIPG Homo sapiens Human PF00151 PF01477 7.4 IC50 ChEMBL;BindingDB