Molecule Details
InChIKeyCKTPSKKTZVSXLI-UHFFFAOYSA-N
Compound Name4-(tert-butyl)-N-(2-oxo-1,2-dihydropyridin-4-yl)-2-((6-(trifluoromethyl)pyridin-3-yl)oxy)benzamide
Canonical SMILESCC(C)(C)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(Oc2ccc(C(F)(F)F)nc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UQD0 SCN8A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 7.1 IC50 ChEMBL;BindingDB
Q9Y5Y9 SCN10A Homo sapiens Human PF00520 PF24609 PF06512 7.1 IC50 ChEMBL;BindingDB