Molecule Details
InChIKeyCKRQXNYHHJWLPU-LECRGTDLSA-N
Compound Name(R)-N-[((S)-1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcarbamoyl)-methyl]-3-(1-carbamimidoyl-piperidin-3-yl)-2-phenylmethanesulfonylamino-propionamide; TFA
Canonical SMILESN=C(N)N1CCCC(C[C@@H](NS(=O)(=O)Cc2ccccc2)C(=O)NCC(=O)N[C@H]2CCCN(C(=N)N)C2O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 9.0 IC50 ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 7.5 IC50 ChEMBL;BindingDB
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 6.1 IC50 ChEMBL;BindingDB