Molecule Details
InChIKeyCKEWXVJUPNKAPF-UHFFFAOYSA-N
Compound Name6-(benzo[d][1,3]dioxol-5-yl)-N-methyl-N-((5-methyl-1,3,4-oxadiazol-2-yl)methyl)quinazolin-4-amine
Canonical SMILESCc1nnc(CN(C)c2ncnc3ccc(-c4ccc5c(c4)OCO5)cc23)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.09
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9HAZ1 CLK4 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
P49759 CLK1 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
Q13627 DYRK1A Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB