Molecule Details
InChIKeyCKASJUOAZZSCTR-UHFFFAOYSA-N
Compound Name1-[4-[1-(2-Fluorophenyl)pyrazolo[4,3-c]pyridin-6-yl]-1-methylpyrazol-5-yl]piperidin-4-amine
Canonical SMILESCn1ncc(-c2cc3c(cn2)cnn3-c2ccccc2F)c1N1CCC(N)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.2
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 7.8 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 7.3 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.5 Ki ChEMBL;BindingDB