Molecule Details
InChIKeyCJXZQDNBKDLDLD-UHFFFAOYSA-N
Compound Name4-N-hydroxy-1-N-[3-[(5-pyridin-3-yl-1,3-thiazol-2-yl)amino]phenyl]benzene-1,4-dicarboxamide
Canonical SMILESO=C(NO)c1ccc(C(=O)Nc2cccc(Nc3ncc(-c4cccnc4)s3)c2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.8
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 7.0 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.7 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.7 pIC50 TTD_MultiTarget