Molecule Details
InChIKeyCJLTWANHPMOFEB-TZIWHRDSSA-N
Compound Name5-N-[(1R,2R)-2-aminocyclohexyl]-3-propan-2-yl-7-N-[(4-pyridin-2-ylphenyl)methyl]-2H-pyrazolo[4,3-d]pyrimidine-5,7-diamine
Canonical SMILESCC(C)c1n[nH]c2c(NCc3ccc(-c4ccccn4)cc3)nc(N[C@@H]3CCCC[C@H]3N)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00535 CDK5 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 7.3 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB