Target not found.
Molecule Details
InChIKeyCJDVFKPJFAFFDM-SNAWJCMRSA-N
Compound NameN-(2-aminophenyl)-5-[[(E)-4-(6-methyl-3-pyridinyl)but-3-enoyl]amino]pyridine-2-carboxamide
Canonical SMILESCc1ccc(/C=C/CC(=O)Nc2ccc(C(=O)Nc3ccccc3N)nc2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O15379 HDAC3 Homo sapiens Human PF00850 8.1 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 7.0 IC50 ChEMBL;BindingDB
Q92769 HDAC2 Homo sapiens Human PF00850 6.4 IC50 ChEMBL;BindingDB