Molecule Details
InChIKeyCHGATQCEUOURQZ-WBXFWKJNSA-N
Canonical SMILESCOc1cc(NC(=O)CCN(C)[C@H]2CC[C@H](OC(=O)C(O)(c3cccs3)c3cccs3)CC2)c(F)cc1CNC[C@H](O)c1ccc(O)c2[nH]c(=O)ccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P20309 CHRM3 Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P07550 ADRB2 Homo sapiens Human PF00001 8.3 IC50 ChEMBL;BindingDB