Molecule Details
InChIKeyCHEUONHPKBJUCB-XMMPIXPASA-N
Compound NamePyrrolidine-1-carboxylic acid (R)-3-oxo-3-(4-phenylcarbamoyl-piperidin-1-yl)-2-(3-m-tolyl-ureido)-propyl ester
Canonical SMILESCc1cccc(NC(=O)N[C@H](COC(=O)N2CCCC2)C(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.47
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 7.5 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 7.5 IC50 ChEMBL;BindingDB