Molecule Details
InChIKeyCHCYABPIGAAURP-UHFFFAOYSA-N
Compound NameN-(azetidin-3-yl)-6-(1-pyridin-2-ylpyrazolo[4,3-c]pyridin-6-yl)pyrazin-2-amine
Canonical SMILESc1ccc(-n2ncc3cnc(-c4cncc(NC5CNC5)n4)cc32)nc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.6 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.4 Ki ChEMBL;BindingDB