Molecule Details
InChIKeyCGHABSNFJJPLNR-UHFFFAOYSA-N
Compound Name2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-N-(4-{2-[8-(4-methyl-piperazin-1-yl)-naphthalen-2-yloxy]-acetylamino}-phenyl)-acetamide
Canonical SMILESCN1CCN(c2cccc3ccc(OCC(=O)Nc4ccc(NC(=O)COc5ccc6[nH]cc(CCN)c6c5)cc4)cc23)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 9.3 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB