Molecule Details
InChIKeyCFTIJALKSHXVNU-QGZVFWFLSA-N
Compound Name(7R)-8-cyclopentyl-2-[2-methoxy-4-(piperidine-1-carbonyl)anilino]-5,7-dimethyl-7H-pteridin-6-one
Canonical SMILESCOc1cc(C(=O)N2CCCCC2)ccc1Nc1ncc2c(n1)N(C1CCCC1)[C@H](C)C(=O)N2C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.0 IC50 ChEMBL;BindingDB
P53350 PLK1 Homo sapiens Human PF00069 PF00659 7.0 IC50 ChEMBL;BindingDB
Q58F21 BRDT Homo sapiens Human PF17035 PF17105 PF00439 6.4 IC50 ChEMBL;BindingDB